Thiorphan

Tiorfan

Engelsk definition

A potent inhibitor of membrane metalloendopeptidase (ENKEPHALINASE). Thiorphan potentiates morphine-induced ANALGESIA and attenuates naloxone-precipitated withdrawal symptoms.

Svenska synonymer

Inga svenska synonymer finns.

Engelska synonymer

(3-Mercapto-2-benzylpropionyl)glycine Tiorphan Thiorphan, (R)-Isomer Thiorphan, (S)-Isomer